SU 5402
Code | Size | Price |
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TAR-T6996-5mg | 5mg | £118.00 | |||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||
Special offer! Add £1 to your order to get a TargetMol CCK-8 Kit. Read more here. |
Quantity:
TAR-T6996-1mL | 1 mL * 10 mM (in DMSO) | £123.00 | |||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||
Special offer! Add £1 to your order to get a TargetMol CCK-8 Kit. Read more here. |
Quantity:
TAR-T6996-10mg | 10mg | £145.00 | |||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||
Special offer! Add £1 to your order to get a TargetMol CCK-8 Kit. Read more here. |
Quantity:
TAR-T6996-25mg | 25mg | £206.00 | |||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||
Special offer! Add £1 to your order to get a TargetMol CCK-8 Kit. Read more here. |
Quantity:
TAR-T6996-50mg | 50mg | £298.00 | |||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||
Special offer! Add £1 to your order to get a TargetMol CCK-8 Kit. Read more here. |
Quantity:
TAR-T6996-100mg | 100mg | £436.00 | |||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||
Special offer! Add £1 to your order to get a TargetMol CCK-8 Kit. Read more here. |
Quantity:
Prices exclude any Taxes / VAT
Overview
Regulatory Status: RUO
Shipping:
cool pack
Storage:
-20℃
Images
Documents
Further Information
Bioactivity:
SU5402 is a potent multi-targeted receptor tyrosine kinase inhibitor with IC50 of 20 nM, 30 nM, and 510 nM for VEGFR2, FGFR1, and PDGF-Rβ, respectively.
CAS:
215543-92-3
Formula:
C17H16N2O3
Molecular Weight:
296.326
Pathway:
Tyrosine Kinase/Adaptors; Angiogenesis
Purity:
0.9964
SMILES:
Cc1c[nH]c(C=C2/C(=O)Nc3ccccc23)c1CCC(O)=O
Target:
VEGFR; FGFR; PDGFR
References
Trzci?ska-Daneluti AM, et al. RNA Interference Screen to Identify Kinases That Suppress Rescue of ?F508-CFTR. Mol Cell Proteomics. 2015 Jun;14(6):1569-83.
Lo AK, et al. J Pathol. 2015. doi: 10.12002/path.4575.
Fong TA, et al. Cancer Res. 1999, 59(1), 99-106.
Sun L, et al. J Med Chem. 1999, 42(25), 5120-5130.
Li Y, et al. Calcif Tissue Int. 2013, 93(6), 556-5 64.