DC260126
Code | Size | Price |
---|
TAR-T7127-5mg | 5mg | £111.00 | |||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||
Special offer! Add £1 to your order to get a TargetMol CCK-8 Kit. Read more here. |
Quantity:
TAR-T7127-1mL | 1 mL * 10 mM (in DMSO) | £114.00 | |||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||
Special offer! Add £1 to your order to get a TargetMol CCK-8 Kit. Read more here. |
Quantity:
TAR-T7127-10mg | 10mg | £124.00 | |||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||
Special offer! Add £1 to your order to get a TargetMol CCK-8 Kit. Read more here. |
Quantity:
TAR-T7127-25mg | 25mg | £186.00 | |||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||
Special offer! Add £1 to your order to get a TargetMol CCK-8 Kit. Read more here. |
Quantity:
TAR-T7127-50mg | 50mg | £253.00 | |||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||
Special offer! Add £1 to your order to get a TargetMol CCK-8 Kit. Read more here. |
Quantity:
Prices exclude any Taxes / VAT
Overview
Regulatory Status: RUO
Shipping:
cool pack
Storage:
-20℃
Images
Documents
Further Information
Bioactivity:
DC260126 is a small-molecule antagonist of FFA1 (GPR40)
CAS:
346692-04-4
Formula:
C16H18FNO2S
Molecular Weight:
307.38
Pathway:
GPCR/G Protein; Apoptosis; Endocrinology/Hormones
Purity:
0.98
SMILES:
CCCCc1ccc(NS(=O)(=O)c2ccc(F)cc2)cc1
Target:
Apoptosis; GPR
References
Peng S , Ting W , Yuren Z , et al. DC260126: A Small-Molecule Antagonist of GPR40 that Protects against Pancreatic ?-Cells Dysfunction in db/db Mice[J]. PLoS ONE, 2013, 8(6):e66744-.
Zhang X , Yan G , Li Y , et al. DC260126, a small-molecule antagonist of GPR40, improves insulin tolerance but not glucose tolerance in obese Zucker rats[J]. Biomedicine and Pharmacotherapy, 2010, 64(9):0-651.