GFT505

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TargetMol
Product Code: TAR-T8699
Supplier: TargetMol
CodeSizePrice
TAR-T8699-5mg5mg£111.00
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Quantity:
TAR-T8699-1mL1 mL * 10 mM (in DMSO)£112.00
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Quantity:
TAR-T8699-10mg10mg£131.00
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Quantity:
TAR-T8699-25mg25mg£173.00
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Quantity:
TAR-T8699-50mg50mg£225.00
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Quantity:
TAR-T8699-100mg100mg£301.00
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Quantity:
TAR-T8699-200mg200mg£417.00
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Quantity:
Prices exclude any Taxes / VAT

Overview

Regulatory Status: RUO
Shipping:
cool pack
Storage:
-20℃

Documents

Further Information

Bioactivity:
GFT505 (Elafibranor) is a PPARα/δ agonist with EC50s of 45 and 175 nM, respectively.
CAS:
824932-88-9
Formula:
C22H24O4S
Molecular Weight:
384.49
Pathway:
DNA Damage/DNA Repair; Metabolism
Purity:
0.9883
SMILES:
CC(C)(C(O)=O)Oc1c(C)cc(C=CC(c(cc2)ccc2SC)=O)cc1C
Target:
PPAR

References

Liu ZM, et al. Early investigational drugs targeting PPAR-? for the treatment of metabolic disease.Expert Opin Investig Drugs. 2015 May;24(5):611-21.