α-Conotoxin PIA
| Code | Size | Price |
|---|
| TAR-TP2065-5mg | 5mg | £1,109.00 | |||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||
| Special offer! Add £1 to your order to get a TargetMol CCK-8 Kit. Read more here. | |||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||
Quantity:
Prices exclude any Taxes / VAT
Overview
Regulatory Status: RUO
Shipping:
cool pack
Storage:
-20℃
Documents
Further Information
Bioactivity:
Selective antagonist of α6-containing nicotinic receptors that discriminates between the closely related α6 and α3 subunits (IC50 values are 0.95 and 74.2 nM for rat α6/α3β2β3 and α3β2 receptors respectively).
CAS:
669050-68-4
Formula:
C79H125N27O25S4
Molecular Weight:
1981.3
Purity:
0.98
SMILES:
0
References
Dowell et al (2003) α-Conotoxin PIA is selective for α6 subunit-containing nicotinic acetylcholine receptors. J.Neurosci. 23 8445 PMID:
Azam and McIntosh (2005) Effect of novel α-Conotoxins on nicotine-stimulated [3H]DA release from rat striatal synaptosomes. J.Pharmacol.Exp.Ther. 312 231 PMID: