Stressin I
Code | Size | Price |
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TAR-TP2125-5mg | 5mg | £969.00 | |||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||
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Overview
Regulatory Status: RUO
Shipping:
cool pack
Storage:
-20℃
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Further Information
Bioactivity:
Potent and selective corticotropin releasing factor receptor-1 (CRF1) agonist (Ki values are 1.5 and 224 nM for CRF1 and CRF2 receptors respectively). Increases ACTH levels and increases faecal pellet output in vivo following i.p. administration.
CAS:
TP2125
Formula:
C203H337N57O56
Molecular Weight:
4472.24
Purity:
0.98
SMILES:
0
References
Rivier et al (2007) Stressin1-A, a potent cortico. releasing factor receptor 1 (CRF1)-selective peptide agonist. J.Med.Chem. 50 1668 PMID:
Rivier et al (2002) Receptor-selective cortico. releasing factor analogs. Endocrin.Soc.Abstr. P2-50 Bruchas et al (2009) CRF1-R activation of the dynorphin/kappa opioid system in the mouse basolateral amygdala mediates anxiety-like behavior. PLoS One. 4 e8528 PMID: