DDR Inhibitor

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TargetMol
Product Code: TAR-T10985
Supplier: TargetMol
CodeSizePrice
TAR-T10985-1mg1mg£230.00
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TAR-T10985-5mg5mg£402.00
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TAR-T10985-1mL1 mL * 10 mM (in DMSO)£436.00
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TAR-T10985-10mg10mg£603.00
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TAR-T10985-25mg25mg£1,139.00
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TAR-T10985-50mg50mg£1,773.00
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TAR-T10985-100mg100mg£2,376.00
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Prices exclude any Taxes / VAT

Overview

Regulatory Status: RUO
Shipping:
cool pack
Storage:
-20℃

Images

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Documents

Further Information

Bioactivity:
DDR inhibitor is a potent discidin domain receptor (DDR) inhibitor. The IC50 of DDR2 is 3.3 nM, and DDR1 has 53% inhibition at 1.5 nM.
CAS:
1644069-80-6
Formula:
C23H20FN5O2
Molecular Weight:
417.44
Pathway:
Tyrosine Kinase/Adaptors
Purity:
0.9775
SMILES:
O=C(NC=1C=CC=C(F)C1)NCC2=CC=C(C(=C2)NC(=O)C3=CN=C4C=CC=CN43)C
Target:
Discoidin Domain Receptor (DDR)

References

1. Gordon Saxty, et al. Imidazo-condensed bicycles as inhibitors of discoidin domain receptors (ddrs)