Penitrem A
| Code | Size | Price |
|---|
| TAR-T12403-10mg | 10mg | £760.00 | |||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||
| Special offer! Add £1 to your order to get a TargetMol CCK-8 Kit. Read more here. | |||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||
Quantity:
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Overview
Regulatory Status: RUO
Shipping:
cool pack
Storage:
-20℃
Documents
Further Information
Bioactivity:
Penitrem A is a selective antagonist of BK channel with antiproliferative and anti-invasive activities against multiple malignancies.
CAS:
12627-35-9
Formula:
C37H44ClNO6
Molecular Weight:
634.21
Purity:
0.98
SMILES:
[H][C@]12C[C@@]3([H])[C@@]1(O)c1c(CC2=C)c(Cl)cc2[nH]c4c(c12)[C@@]([H])(OC3(C)C)[C@]1([H])CC[C@@]2(O)[C@@]35O[C@@H]3[C@@H](O)[C@H](O[C@@]5([H])CC[C@]2(C)[C@@]41C)C(C)=C
References
1. Goda AA, et al. The Maxi-K (BK) Channel Antagonist Penitrem A as a Novel Breast Cancer-Targeted Therapeutic. Mar Drugs. 2018 May 11;16(5).
2. Norris PJ, et al. Actions of tremorgenic fungal toxins on neurotransmitter release. J Neurochem. 1980 Jan;34(1):33-42.