TR antagonist 1
Code | Size | Price |
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TAR-T13435-5mg | 5mg | £437.00 | |||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||
Special offer! Add £1 to your order to get a TargetMol CCK-8 Kit. Read more here. |
Quantity:
TAR-T13435-50mg | 50mg | £1,765.00 | |||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||
Special offer! Add £1 to your order to get a TargetMol CCK-8 Kit. Read more here. |
Quantity:
TAR-T13435-100mg | 100mg | £2,697.00 | |||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||
Special offer! Add £1 to your order to get a TargetMol CCK-8 Kit. Read more here. |
Quantity:
Prices exclude any Taxes / VAT
Overview
Regulatory Status: RUO
Shipping:
cool pack
Storage:
-20℃
Images
Documents
Further Information
Bioactivity:
TR antagonist 1 is a high-affinity antagonist of thyroid hormone receptor (TR) (IC50s of 36 and 22 nM for TRα and TRβ, respectively).
CAS:
500794-88-7
Formula:
C25H23Br2NO4
Molecular Weight:
561.27
Purity:
0.98
SMILES:
CC(C)c1cc(Oc2c(Br)cc(CCC(O)=O)cc2Br)cc(C=Cc2ccncc2)c1O
References
1. Koehler K, et al. Thyroid receptor ligands. 6. A high affinity "direct antagonist" selective for the thyroid hormone receptor. J Med Chem. 2006 Nov 16;49(23):6635-7.