HIF-2 α-IN-1
Code | Size | Price |
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TAR-T15482-5mg | 5mg | £850.00 | |||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||
Special offer! Add £1 to your order to get a TargetMol CCK-8 Kit. Read more here. |
Quantity:
TAR-T15482-50mg | 50mg | £1,830.00 | |||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||
Special offer! Add £1 to your order to get a TargetMol CCK-8 Kit. Read more here. |
Quantity:
TAR-T15482-100mg | 100mg | £2,560.00 | |||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||
Special offer! Add £1 to your order to get a TargetMol CCK-8 Kit. Read more here. |
Quantity:
Prices exclude any Taxes / VAT
Overview
Regulatory Status: RUO
Shipping:
cool pack
Storage:
-20℃
Images
Documents
Further Information
Bioactivity:
HIF-2α-IN-1 is an inhibitor of HIF-2α. In HIF-2α scintillation proximity assay, It also has an IC50 of less than 500 nM.
CAS:
1799948-06-3
Formula:
C16H8F5NO4S
Molecular Weight:
405.3
Purity:
0.98
SMILES:
O[C@@H]1c2c(ccc(Oc3cc(F)cc(c3)C#N)c2C(F)F)S(=O)(=O)C1(F)F
References
1. Bruick Richard Keith, et al. HIF-2? inhibitors for treating iron overload disorders. From PCT Int. Appl. (2016), WO 2016057242 A1 20160414.
2. Dixon Darryl David, et al. Preparation of cyclic sulfone and sulfoximine analogs as HIF-2? inhibitors. From PCT Int. Appl. (2015), WO 2015095048 A1 20150625.