TargetMol

Mubritinib

Product Code:
 
TAR-T6124
Product Group:
 
Inhibitors and Activators
Supplier:
 
TargetMol
Regulatory Status:
 
RUO
Shipping:
 
cool pack
Storage:
 
-20℃
1 / 1
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CodeSizePrice
TAR-T6124-1mL1 mL * 10 mM (in DMSO)£111.00
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TAR-T6124-10mg10mg£114.00
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TAR-T6124-25mg25mg£152.00
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TAR-T6124-50mg50mg£207.00
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TAR-T6124-100mg100mg£324.00
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TAR-T6124-200mg200mg£495.00
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This product comes from: United States.
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Further Information

Bioactivity:
Mubritinib (TAK-165) is a potent inhibitor of HER2/ErbB2 with IC50 of 6 nM.
CAS:
366017-09-6
Formula:
C25H23F3N4O2
Molecular Weight:
468.48
Pathway:
Chromatin/Epigenetic; Stem Cells; JAK/STAT signaling; Tyrosine Kinase/Adaptors; Angiogenesis
Purity:
0.9957
SMILES:
FC(F)(F)c1ccc(C=Cc2nc(COc3ccc(CCCCn4ccnn4)cc3)co2)cc1
Target:
EGFR; FGFR; JAK; PDGFR

References

Nagasawa J, et al. Int J Urol, 2006, 13(5), 587-592.