Salirasib
Code | Size | Price |
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TAR-T6163-10mg | 10mg | £111.00 | |||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||
Special offer! Add £1 to your order to get a TargetMol CCK-8 Kit. Read more here. |
Quantity:
TAR-T6163-25mg | 25mg | £149.00 | |||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||
Special offer! Add £1 to your order to get a TargetMol CCK-8 Kit. Read more here. |
Quantity:
TAR-T6163-50mg | 50mg | £201.00 | |||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||
Special offer! Add £1 to your order to get a TargetMol CCK-8 Kit. Read more here. |
Quantity:
TAR-T6163-100mg | 100mg | £258.00 | |||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||
Special offer! Add £1 to your order to get a TargetMol CCK-8 Kit. Read more here. |
Quantity:
TAR-T6163-200mg | 200mg | £389.00 | |||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||
Special offer! Add £1 to your order to get a TargetMol CCK-8 Kit. Read more here. |
Quantity:
Prices exclude any Taxes / VAT
Overview
Regulatory Status: RUO
Shipping:
cool pack
Storage:
-20℃
Images
Documents
Further Information
Bioactivity:
Salirasib(Ki=2.6 μM), an effective competitive prenylated protein methyltransferase (PPMTase) inhibitor, inhibits Ras methylation with potential antineoplastic activity.
CAS:
162520-00-5
Formula:
C22H30O2S
Molecular Weight:
358.54
Pathway:
Autophagy; MAPK; GPCR/G Protein
Purity:
0.9933
SMILES:
CC(C)=CCCC(C)=CCCC(C)=CCSc1ccccc1C(O)=O
Target:
Autophagy; Ras
References
Gana-Weisz M, et al. Biochem Biophys Res Commun. 1997, 900-904.
Marciano D, et al. J Med Chem. 1995, 38(8), 1267-1272.
Marom M, et al. J Biol Chem. 1995, 270(38), 22263-22270.
Reif S, et al. J Hepatol. 1999, 31(6),, 1053-1061.
Weisz B, et al. Oncogene. 1999, 18(16), 2579-2588.