(R)-PS210
Code | Size | Price |
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TAR-T12639-50mg | 50mg | £870.00 | |||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||
Special offer! Add £1 to your order to get a TargetMol CCK-8 Kit. Read more here. |
Quantity:
TAR-T12639-100mg | 100mg | £1,364.00 | |||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||
Special offer! Add £1 to your order to get a TargetMol CCK-8 Kit. Read more here. |
Quantity:
Prices exclude any Taxes / VAT
Overview
Regulatory Status: RUO
Shipping:
cool pack
Storage:
-20℃
Images
Documents
Further Information
Bioactivity:
(R)-PS210, the R enantiomer of PS210 is a substrate-selective allosteric PDK1 activator with an (AC50 of 1.8 μM).
CAS:
1410101-89-1
Formula:
C19H15F3O5
Molecular Weight:
380.319
Purity:
0.98
SMILES:
OC(=O)C([C@@H](CC(=O)c1ccc(cc1)C(F)(F)F)c1ccccc1)C(O)=O
References
1. Wilhelm A, et al. 2-(3-Oxo-1,3-diphenylpropyl)malonic?acids?as?potent?allosteric?ligands?of the?PIF?pocket?of?phosphoinositide-dependent?kinase-1:?development?and?prodrug?concept.J Med Chem.?2012 Nov 26;55(22):9817-30.