Tilfrinib

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TargetMol
Product Code: TAR-T17098
Supplier: TargetMol
CodeSizePrice
TAR-T17098-1mg1mg£101.00
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TAR-T17098-2mg2mg£114.00
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TAR-T17098-1mL1 mL * 10 mM (in DMSO)£142.00
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TAR-T17098-5mg5mg£142.00
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TAR-T17098-10mg10mg£182.00
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TAR-T17098-25mg25mg£287.00
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TAR-T17098-50mg50mg£462.00
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TAR-T17098-100mg100mg£646.00
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TAR-T17098-500mg500mg£1,259.00
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Prices exclude any Taxes / VAT

Overview

Regulatory Status: RUO
Shipping:
cool pack
Storage:
-20℃

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Documents

Further Information

Bioactivity:
Tilfrinib is an effective and selective inhibitor of breast tumor kinase(Brk, IC50 = 3.15 nM) which displays anti-proliferative and anti-tumor activities.
CAS:
1600515-49-8
Formula:
C17H13N3O
Molecular Weight:
275.3
Pathway:
Angiogenesis; Tyrosine Kinase/Adaptors
Purity:
0.9973
SMILES:
OC1=CC=CC(=C1)NC2=CC=NC=3NC=4C=CC=CC4C32
Target:
BTK

References

Mahmoud KA, et al. Discovery of 4-anilino ?-carbolines as novel Brk inhibitors. Bioorg Med Chem Lett. 2014 Apr 15;24(8):1948-51. Mahmoud KA, et al. Discovery of 4-anilino ?-carbolines as novel Brk inhibitors. Bioorg Med Chem Lett. 2014 Apr 15;24(8):1948-51.