GSK 591 dihydrochloride

TargetMol
Product Code: TAR-T36981
Supplier: TargetMol
CodeSizePrice
TAR-T36981-25mg25mg£922.00
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Overview

Regulatory Status: RUO
Shipping:
cool pack
Storage:
-20℃

Images

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Further Information

Bioactivity:
Potent and selective PRMT5 inhibitor (IC50 = 4 nM). Selective for PRMT5 over a panel of other PRMTs and lysine methyltransferases. Inhibits proliferation of mantle cell lymphoma (MCL) in vitro. To request the negative control for GSK 591, please fill out the SGC 2096 request form on the SGC website.
CAS:
2320953-89-5
Formula:
C22H28N4O2.2HCl
Molecular Weight:
453.41
Purity:
0.98
SMILES:
O[C@@H](CNC(C1=CC=NC(NC2CCC2)=C1)=O)CN3CC4=CC=CC=C4CC3.Cl.Cl