Linagliptin
Code | Size | Price |
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TAR-T0191-50mg | 50mg | £101.00 | |||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||
Special offer! Add £1 to your order to get a TargetMol CCK-8 Kit. Read more here. |
Quantity:
TAR-T0191-1mL | 1 mL * 10 mM (in DMSO) | £111.00 | |||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||
Special offer! Add £1 to your order to get a TargetMol CCK-8 Kit. Read more here. |
Quantity:
TAR-T0191-100mg | 100mg | £114.00 | |||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||
Special offer! Add £1 to your order to get a TargetMol CCK-8 Kit. Read more here. |
Quantity:
Prices exclude any Taxes / VAT
Overview
Regulatory Status: RUO
Shipping:
cool pack
Storage:
-20℃
Images
Documents
Further Information
Bioactivity:
Linagliptin is a potent, orally bioavailable dihydropurinedione-based inhibitor of dipeptidyl peptidase 4 (DPP-4), with hypoglycemic activity.
CAS:
668270-12-0
Formula:
C25H28N8O2
Molecular Weight:
472.553
Pathway:
Proteases/Proteasome; Cell Cycle/Checkpoint; Ubiquitination; Autophagy; Apoptosis
Purity:
0.9995
SMILES:
CC#CCn1c(nc2n(C)c(=O)n(Cc3nc(C)c4ccccc4n3)c(=O)c12)N1CCC[C@@H](N)C1
Target:
Ferroptosis; Proteasome; DPP-4; Autophagy
References
1. Eckhardt M, et al. J Med Chem. 2007, 50(26), 6450-6453.
2. Thomas L, J Pharmacol Exp Ther. 2008, 325(1), 175-182.
3. Sch?rmann C, et al. J Pharmacol Exp Ther. 2012, 342(1), 71-8.