(5Z,2E)-CU-3
Code | Size | Price |
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TAR-T10177-100mg | 100mg | Enquire | |||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||
Special offer! Add £1 to your order to get a TargetMol CCK-8 Kit. Read more here. |
Quantity:
TAR-T10177-50mg | 50mg | Enquire | |||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||
Special offer! Add £1 to your order to get a TargetMol CCK-8 Kit. Read more here. |
Quantity:
Prices exclude any Taxes / VAT
Overview
Regulatory Status: RUO
Shipping:
cool pack
Storage:
-20℃
Images
Documents
Further Information
Bioactivity:
(5Z,2E)-CU-3 is a selective inhibitor against the α-isozyme of DGK (IC50: 0.6 μM), competitively inhibits the affinity of DGKα for ATP (Km: 0.48 mM).
CAS:
1815598-71-0
Formula:
C16H12N2O4S3
Molecular Weight:
392.47
Purity:
0.98
SMILES:
O=S(C1=CC=CC=C1)(NN(C/2=O)C(SC2=C/C=C/C3=CC=CO3)=S)=O
References
1. Liu K, et al. A novel diacylglycerol kinase ?-selective inhibitor, CU-3, induces cancer cell apoptosis and enhances immune response. J Lipid Res. 2016 Mar;57(3):368-79.