Deltasonamide 2 (TFA)
Code | Size | Price |
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TAR-T10994L2-5mg | 5mg | £304.00 | |||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||
Special offer! Add £1 to your order to get a TargetMol CCK-8 Kit. Read more here. |
Quantity:
TAR-T10994L2-50mg | 50mg | £1,163.00 | |||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||
Special offer! Add £1 to your order to get a TargetMol CCK-8 Kit. Read more here. |
Quantity:
TAR-T10994L2-100mg | 100mg | £1,830.00 | |||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||
Special offer! Add £1 to your order to get a TargetMol CCK-8 Kit. Read more here. |
Quantity:
Prices exclude any Taxes / VAT
Overview
Regulatory Status: RUO
Shipping:
cool pack
Storage:
-20℃
Images
Documents
Further Information
Bioactivity:
Deltasonamide 2 TFA is competitive, high affinity PDEδ inhibitor with a Kd of ~385 pM.
CAS:
2235358-74-2
Formula:
C32H40ClF3N6O6S2
Molecular Weight:
761.27
Pathway:
Metabolism
Purity:
0.98
SMILES:
OC(=O)C(F)(F)F.CNc1nccc(CN([C@H]2CC[C@H](N)CC2)S(=O)(=O)c2ccc(cc2)S(=O)(=O)N(Cc2ccc(Cl)cc2)C2CCCC2)n1
Target:
PDE
References
1. Klein CH, et al. PDE? inhibition impedes the proliferation and survival of human colorectal cancer cell linesharboring oncogenic KRas. Int J Cancer. 2019 Feb 15;144(4):767-776.