0990CL

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TargetMol
Product Code: TAR-T13983
Supplier: TargetMol
CodeSizePrice
TAR-T13983-1mg1mg£242.00
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TAR-T13983-5mg5mg£503.00
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Quantity:
TAR-T13983-1mL1 mL * 10 mM (in DMSO)£523.00
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Quantity:
TAR-T13983-10mg10mg£695.00
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Quantity:
TAR-T13983-25mg25mg£1,018.00
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TAR-T13983-50mg50mg£1,372.00
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Quantity:
TAR-T13983-100mg100mg£1,821.00
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Prices exclude any Taxes / VAT

Overview

Regulatory Status: RUO
Shipping:
cool pack
Storage:
-20℃

Images

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Documents

Further Information

Bioactivity:
0990CL is able to block α2AR mediated regulation of cAMP. 0990CL is a specific heterotrimeric Gαi subunit inhibitor by direct interaction with Gαi.
CAS:
511514-03-7
Formula:
C21H21N5
Molecular Weight:
343.434
Pathway:
GPCR/G Protein|Others
Purity:
0.98
SMILES:
CC1=CC(C)(C)N=C(Nc2nc(-c3ccccc3)c3ccccc3n2)N1
Target:
Others|cAMP

References

1. Appleton KM,et al. Development of inhibitors of heterotrimeric G?i subunits.Bioorg Med Chem. 2014 Jul 1;22(13):3423-34.