TargetMol

Ajmaline

Product Code:
 
TAR-T4550
Supplier:
 
TargetMol
Regulatory Status:
 
RUO
Shipping:
 
cool pack
Storage:
 
-20℃
1 / 1
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CodeSizePrice
TAR-T4550-50mg50mg£103.00
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Quantity:
TAR-T4550-1mL1 mL * 10 mM (in DMSO)£107.00
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Quantity:
TAR-T4550-100mg100mg£124.00
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Further Information

Bioactivity:
Ajmaline is a class Ia anti-arrhythmic compound that is widely used for the diagnosis of Brugada syndrome and the acute treatment of atrial or ventricular tachycardia. Ajmaline inhibits cardiac Kv1.5 and Kv4.3 channels at therapeutic concentrations.
CAS:
4360-12-7
Formula:
C20H26N2O2
Molecular Weight:
326.44
Pathway:
Membrane transporter/Ion channel
Purity:
0.9967
SMILES:
CC[C@H]1[C@@H]2C[C@H]3[C@@H]4N(C)c5ccccc5[C@]44C[C@@H](C2[C@H]4O)N3[C@@H]1O
Target:
Sodium Channel

References

Fischer F, et al. Inhibition of cardiac Kv1.5 and Kv4.3 potassium channels by the class Ia anti-arrhythmic ajmaline: mode of action.[J]. Naunyn-Schmiedeberg's Archives of Pharmacology, 2013, 386(11):991-999.