M77976

TargetMol
Product Code: TAR-T15944
Supplier: TargetMol
CodeSizePrice
TAR-T15944-100mg100mgEnquire
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TAR-T15944-50mg50mgEnquire
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Overview

Regulatory Status: RUO
Shipping:
cool pack
Storage:
-20℃

Images

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Further Information

Bioactivity:
M77976 is the potential for the research of obesity and diabetes. M77976 is a specific ATP-competitive inhibitor of PDK4 (pyruvate dehydrogenase kinase isoforms 4) (IC50: 648 μM).
CAS:
394237-61-7
Formula:
C17H16N2O3
Molecular Weight:
296.326
Pathway:
Neuroscience
Purity:
0.98
SMILES:
COc1ccc(cc1)-c1c(C)[nH]nc1-c1ccc(O)cc1O
Target:
GluR

References

1. Kukimoto-Niino M, et al. Inhibitor-bound structures of human pyruvate dehydrogenase kinase 4. Acta Crystallogr D Biol Crystallogr. 2011 Sep;67(Pt 9):763-73.