TargetMol

M77976

Product Code:
 
TAR-T15944
Product Group:
 
Inhibitors and Activators
Supplier:
 
TargetMol
Regulatory Status:
 
RUO
Shipping:
 
cool pack
Storage:
 
-20℃
1 / 1
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Further Information

Bioactivity:
M77976 is the potential for the research of obesity and diabetes. M77976 is a specific ATP-competitive inhibitor of PDK4 (pyruvate dehydrogenase kinase isoforms 4) (IC50: 648 μM).
CAS:
394237-61-7
Formula:
C17H16N2O3
Molecular Weight:
296.326
Pathway:
Neuroscience
Purity:
0.98
SMILES:
COc1ccc(cc1)-c1c(C)[nH]nc1-c1ccc(O)cc1O
Target:
GluR

References

1. Kukimoto-Niino M, et al. Inhibitor-bound structures of human pyruvate dehydrogenase kinase 4. Acta Crystallogr D Biol Crystallogr. 2011 Sep;67(Pt 9):763-73.