Picrotin

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TargetMol
Product Code: TAR-T16533
Supplier: TargetMol
CodeSizePrice
TAR-T16533-1mg1mg£102.00
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TAR-T16533-1mL1 mL * 10 mM (in DMSO)£182.00
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TAR-T16533-5mg5mg£185.00
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TAR-T16533-10mg10mg£230.00
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TAR-T16533-25mg25mg£357.00
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TAR-T16533-50mg50mg£495.00
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TAR-T16533-100mg100mg£678.00
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TAR-T16533-500mg500mg£1,299.00
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Prices exclude any Taxes / VAT

Overview

Regulatory Status: RUO
Shipping:
cool pack
Storage:
-20℃

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Documents

Further Information

Bioactivity:
Picrotin is an inhibitor of glycine receptors. Picrotin blocks α2 GlyR, α1 GlyR and α3 GlyR.
CAS:
21416-53-5
Formula:
C15H18O7
Molecular Weight:
310.302
Pathway:
Membrane transporter/Ion channel
Purity:
0.98
SMILES:
[H][C@@]12OC(=O)[C@@]([H])([C@]1([H])C(C)(C)O)[C@]1(O)C[C@H]3O[C@]33C(=O)O[C@@]2([H])[C@]13C
Target:
Chloride channel

References

1. Li P, et al. Gating effects on picrotin block of glycine receptors. Neuroreport. 2012 Dec 5;23(17):1017-20. 2. Yang Z, et al. A proposed structural basis for picrotoxinin and picrotin binding in the glycine receptor pore. J Neurochem. 2007 Oct;103(2):580-9.