Afloqualone

TargetMol
Product Code: TAR-T4993
Supplier: TargetMol
CodeSizePrice
TAR-T4993-100mg100mg£115.00
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Quantity:
TAR-T4993-1mL1 mL * 10 mM (in DMSO)£119.00
Special offer! Add £1 to your order to get a TargetMol CCK-8 Kit. Read more here.
Quantity:
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Overview

Regulatory Status: RUO
Shipping:
cool pack
Storage:
-20℃

Images

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Further Information

Bioactivity:
Afloqualone is a agonist of GABA receptor . Target: GABA Receptor in vitro: Afloqualone is a quinazolinone family GABAergic drug. Afloqualone is an analogue of methaqualone. It has sedative and muscle-relaxant effects, resulting from its agonist activity at the β subtype of the GABAa receptor.
CAS:
56287-74-2
Formula:
C16H14FN3O
Molecular Weight:
283.306
Pathway:
Membrane transporter/Ion channel; Neuroscience
Purity:
0.9972
SMILES:
Cc1ccccc1-n1c(CF)nc2ccc(N)cc2c1=O
Target:
GABA Receptor

References

Yamamura M, et al. Effects of afloqualone, a new centrally acting muscle relaxant, on DRL response and CER in rats (author's transl). Nihon Yakurigaku Zasshi. 1981 Oct;78(4):381-92.