TargetMol

Proxyphylline

Product Code:
 
TAR-T5940
Supplier:
 
TargetMol
Regulatory Status:
 
RUO
Shipping:
 
cool pack
Storage:
 
-20℃
1 / 1
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CodeSizePrice
TAR-T5940-500mg500mg£103.00
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Quantity:
TAR-T5940-1mL1 mL * 10 mM (in DMSO)£107.00
Special offer! Add £1 to your order to get a TargetMol CCK-8 Kit. Read more here.
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Further Information

Bioactivity:
Proxyphylline is a dual of adenosine A1/A2a receptor inhibitor and phosphodiesterase (PDE) inhibitor. Proxyphylline acts as a cardiac stimulant, vasodilator and bronchodilator.
CAS:
603-00-9
Formula:
C10H14N4O3
Molecular Weight:
238.247
Pathway:
GPCR/G Protein; Metabolism; Neuroscience
Purity:
0.9979
SMILES:
CC(O)Cn1cnc2n(C)c(=O)n(C)c(=O)c12
Target:
PDE; Adenosine Receptor

References

Kukovetz W R , G P?ch, Holzmann S . Overadditive synergism between theophylline, diprophylline and proxyphylline in tracheal smooth muscle relaxation[J]. Arzneimittel-Forschung, 1983, 33(10):1450-1454. Rasmussen F V , Waldorff S , Madsen L . Pharmacokinetics and bronchodilatory effect of proxyphylline and theophylline.[J]. Eur J Respir Dis, 1984, 65(1):20-27. Takeda K , Katano Y , Nakagawa Y , et al. EFFECTS OF AMINOPHYLLINE, PROXYPHYLLINE AND A PROXYPHYLLINE-MELILOTUS EXTRACT-RUTIN MIXTURE (THEOESBERIVEN) ON THE HEART AND THE CORONARY CIRCULATION[J]. The Japanese Journal of Pharmacology, 1977, 27(5):709-720.