BLU0588

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TargetMol
Product Code: TAR-T60169
Supplier: TargetMol
CodeSizePrice
TAR-T60169-1mg1mg£227.00
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TAR-T60169-5mg5mg£430.00
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TAR-T60169-1mL1 mL * 10 mM (in DMSO)£470.00
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TAR-T60169-10mg10mg£599.00
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TAR-T60169-25mg25mg£863.00
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Quantity:
TAR-T60169-50mg50mg£1,179.00
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Quantity:
TAR-T60169-100mg100mg£1,589.00
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TAR-T60169-500mg500mg£3,107.00
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Quantity:
Prices exclude any Taxes / VAT

Overview

Regulatory Status: RUO
Shipping:
cool pack
Storage:
-20°C

Images

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Documents

Further Information

Bioactivity:
BLU0588 is a selective PRKACA inhibitor. BLU0588 inhibits PRKACA catalytic activity with a half-maximal inhibitory concentration (IC50) of 1 nM.
CAS:
T60169
Formula:
C26H25N5O
Molecular Weight:
423.51
Purity:
0.9825
SMILES:
O=C(N[C@@H]1C2=C(C=CC=C2)C[C@H]1N1CCCC1)C1=CC=C(C2=C3C=CNC3=NC=C2)N=C1

References

Stefanie S. Schalm, et al. Evaluation of PRKACA as a Therapeutic Target for Fibrolamellar Carcinoma. bioRxiv 2022.01.31.477690.