TargetMol

CQ211

Product Code:
 
TAR-T63642
Product Group:
 
Inhibitors and Activators
Supplier:
 
TargetMol
Regulatory Status:
 
RUO
Shipping:
 
cool pack
Storage:
 
-20°C
1 / 1
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CodeSizePrice
TAR-T63642-1mg1mg£352.00
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Quantity:
TAR-T63642-5mg5mg£736.00
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Quantity:
TAR-T63642-10mg10mg£978.00
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Quantity:
TAR-T63642-25mg25mg£1,348.00
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Quantity:
TAR-T63642-50mg50mg£1,661.00
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Quantity:
TAR-T63642-100mg100mg£2,079.00
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Quantity:
TAR-T63642-500mg500mg£4,006.00
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This product comes from: United States.
Typical lead time: 10-14 working days.
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Further Information

Bioactivity:
CQ211 is a potent and selective RIOK2 inhibitor with a Kd of 6.1 nM.CQ211 has shown potent proliferation inhibitory activity against various cancer cell lines in vitro.
CAS:
2648986-65-4
Molecular Weight:
521.49
Purity:
0.9701
SMILES:
O=C1NC2=CC=C(C=C2C3=C1N=NN3C4=CC=C(C(=C4)C(F)(F)F)N5CCNCC5)C=6C=NC(OC)=CC6

References

Ouyang Y, et al. Discovery of 8-(6-Methoxypyridin-3-yl)-1-(4-(piperazin-1-yl)-3-(trifluoromethyl)phenyl)-1,5-dihydro-4H-[1,2,3]triazolo[4,5-c]quinolin-4-one (CQ211) as a Highly Potent and Selective RIOK2 Inhibitor. J Med Chem. 2022;65(11):7833-7842.