TargetMol

Eggmanone

Product Code:
 
TAR-T22077
Product Group:
 
Inhibitors and Activators
Supplier:
 
TargetMol
Regulatory Status:
 
RUO
Shipping:
 
cool pack
Storage:
 
-20°C
1 / 1

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CodeSizePrice
TAR-T22077-5mg5mg£850.00
Special offer! Add £1 to your order to get a TargetMol CCK-8 Kit. Read more here.
Quantity:
TAR-T22077-50mg50mg£1,661.00
Special offer! Add £1 to your order to get a TargetMol CCK-8 Kit. Read more here.
Quantity:
TAR-T22077-100mg100mg£2,079.00
Special offer! Add £1 to your order to get a TargetMol CCK-8 Kit. Read more here.
Quantity:
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This product comes from: United States.
Typical lead time: 10-14 working days.
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Further Information

Bioactivity:
Eggmanone (EGM1) is a potent and selective phosphodiesterase 4 (PDE4) antagonist with an IC 50 of 72 nM for PDE4D3. Eggmanone exhibits approximately 40- to 50-fold selective for PDE4D3 over other PDEs. Eggmanone exerts its Hh-inhibitory effects by selective antagonism of PDE4, leading to protein kinase A activation and subsequent Hh blockade [1].
CAS:
505068-32-6
Molecular Weight:
416.58
Purity:
0.98
SMILES:
O=C1C2=C(N=C(SCC(=O)C=3SC=CC3)N1CC(=C)C)SC4=C2CCCC4