LDHA/PDKs-IN-1
Code | Size | Price |
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TAR-T61339-5mg | 5mg | £1,167.00 | |||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||
Special offer! Add £1 to your order to get a TargetMol CCK-8 Kit. Read more here. |
Quantity:
TAR-T61339-50mg | 50mg | £2,307.00 | |||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||
Special offer! Add £1 to your order to get a TargetMol CCK-8 Kit. Read more here. |
Quantity:
TAR-T61339-100mg | 100mg | £2,898.00 | |||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||
Special offer! Add £1 to your order to get a TargetMol CCK-8 Kit. Read more here. |
Quantity:
Prices exclude any Taxes / VAT
Overview
Regulatory Status: RUO
Shipping:
cool pack
Storage:
-20°C
Images
Documents
Further Information
Bioactivity:
LDHA/PDKs-IN-1 (compound 20e) is a highly effective dual inhibitor of PDKs and LDHA, displaying IC50 values of 0.8 uM and 0.15 uM, respectively. It significantly suppresses A549 cell proliferation (EC50 = 13.2 uM), reduces lactate formation, and enhances oxygen consumption. This compound holds great promise for cancer research [1].
CAS:
2490699-40-4
Formula:
C19H21FN2O4
Molecular Weight:
360.385
Purity:
0.98
SMILES:
Cc1occc(=O)c1OCCN1CCN(CC1)C(=O)c1ccc(F)cc1