LSD1-IN-20
Code | Size | Price |
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TAR-T63140-5mg | 5mg | £850.00 | |||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||
Special offer! Add £1 to your order to get a TargetMol CCK-8 Kit. Read more here. |
Quantity:
TAR-T63140-50mg | 50mg | £1,661.00 | |||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||
Special offer! Add £1 to your order to get a TargetMol CCK-8 Kit. Read more here. |
Quantity:
TAR-T63140-100mg | 100mg | £2,079.00 | |||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||
Special offer! Add £1 to your order to get a TargetMol CCK-8 Kit. Read more here. |
Quantity:
Prices exclude any Taxes / VAT
Overview
Regulatory Status: RUO
Shipping:
cool pack
Storage:
-20°C
Images
Documents
Further Information
Bioactivity:
LSD1-IN-20 (compound 1) is a potent, noncovalent, and dual LSD1 (Ki: 0.44 uM), G9a (Ki: 0.68 uM) inhibitor. LSD1-IN-20 could inhibit the proliferation of THP-1 leukemia cells and MDA-MB-231 breast cancer cells, and its 72h IC50 values were 0.51 and 1.60 uM, respectively.
CAS:
1239589-91-3
Molecular Weight:
478.641
Purity:
0.98
SMILES:
COc1cc2nc(NCCCN(C)C)nc(NC3CCN(Cc4ccccc4)CC3)c2cc1OC