HDAC/Top-IN-1
Code | Size | Price |
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TAR-T63543-5mg | 5mg | £1,167.00 | |||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||
Special offer! Add £1 to your order to get a TargetMol CCK-8 Kit. Read more here. |
Quantity:
TAR-T63543-50mg | 50mg | £2,307.00 | |||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||
Special offer! Add £1 to your order to get a TargetMol CCK-8 Kit. Read more here. |
Quantity:
TAR-T63543-100mg | 100mg | £2,898.00 | |||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||
Special offer! Add £1 to your order to get a TargetMol CCK-8 Kit. Read more here. |
Quantity:
Prices exclude any Taxes / VAT
Overview
Regulatory Status: RUO
Shipping:
cool pack
Storage:
-20°C
Images
Documents
Further Information
Bioactivity:
HDAC/Top-IN-1 is a broad-spectrum, orally active dual HDAC/Top inhibitor that acts on HDAC1 (IC50: 0.036 uM), HDAC2 (IC50: 0.14 uM), HDAC3 (IC50: 0.059 uM), HDAC6 (IC50: 0.089 uM) and HDAC8 ( IC50: 9.8 uM). HDAC/Top-IN-1 was able to block HEL cells in S-phase and effectively induce apoptosis.
CAS:
2411379-14-9
Molecular Weight:
512.541
Purity:
0.98
SMILES:
CN1C2N(CCc3c2[nH]c2ccc(OCc4ccc(\C=C\C(=O)NO)cc4)cc32)C(=O)c2cc(F)ccc12