Relutrigine
Code | Size | Price |
---|
TAR-T69652-5mg | 5mg | £930.00 | |||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||
Special offer! Add £1 to your order to get a TargetMol CCK-8 Kit. Read more here. |
Quantity:
TAR-T69652-50mg | 50mg | £1,821.00 | |||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||
Special offer! Add £1 to your order to get a TargetMol CCK-8 Kit. Read more here. |
Quantity:
TAR-T69652-100mg | 100mg | £2,319.00 | |||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||
Special offer! Add £1 to your order to get a TargetMol CCK-8 Kit. Read more here. |
Quantity:
Prices exclude any Taxes / VAT
Overview
Regulatory Status: RUO
Shipping:
cool pack
Storage:
-20°C
Images
Documents
Further Information
Bioactivity:
Relutrigine (PRAX-562) is an orally active inhibitor of persistent sodium channel . Relutrigine potently and preferentially inhibits persistent I Na induced by ATX-II (Nav 1.5 activator) or the SCN8A mutation N1768D with IC 50 values of 141 nM and 75 nM, respectively. Relutrigine exhibits potent use-dependent block and reduces neuronal intrinsic excitability. Relutrigine has effective anticonvulsant activity .
CAS:
2392951-29-8
Molecular Weight:
407.27
Purity:
0.98
SMILES:
FC=1C=C(C=NC1OCC(F)(F)F)C=2N=CC3=NN=C(N3C2)C(F)(F)OCC