PROTAC AR-V7 degrader-1
Code | Size | Price |
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TAR-T74410-50mg | 50mg | Enquire | |||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||
Special offer! Add £1 to your order to get a TargetMol CCK-8 Kit. Read more here. |
Quantity:
TAR-T74410-5mg | 5mg | Enquire | |||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||
Special offer! Add £1 to your order to get a TargetMol CCK-8 Kit. Read more here. |
Quantity:
Prices exclude any Taxes / VAT
Overview
Regulatory Status: RUO
Shipping:
cool pack
Storage:
-20°C
Documents
Further Information
Bioactivity:
PROTAC AR-V7 degrader-1 (Compound 6) is a potent, orally?bioavailable and selective AR-V7 degrader with the DC 50 of 0.32?uM by recruiting VHL E3?ligase?to Androgen receptor?(AR) DNA binding?domain (DBD) binder. PROTAC AR-V7 degrader-1 exhibits activity against 22Rv1 cell-line expressing AR-V7 with the EC 50 of 0.88 uM [1] .
CAS:
2767440-24-2
Molecular Weight:
789.02
Purity:
0.98