ITK degrader 1
Code | Size | Price |
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TAR-T74843-50mg | 50mg | Enquire | |||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||
Special offer! Add £1 to your order to get a TargetMol CCK-8 Kit. Read more here. |
Quantity:
TAR-T74843-5mg | 5mg | Enquire | |||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||
Special offer! Add £1 to your order to get a TargetMol CCK-8 Kit. Read more here. |
Quantity:
Prices exclude any Taxes / VAT
Overview
Regulatory Status: RUO
Shipping:
cool pack
Storage:
-20°C
Documents
Further Information
Bioactivity:
ITK degrader 1 is a highly selective degrader of interleukin-2-inducible T-cell kinase ( ITK ; DC 50 =3.6 nM in vivo in mice). ITK degrader 1 induces rapid, and prolonged ITK degradation and suppresses IL-2 secretion ( EC 50 =35.2 nM, Jurkat cells) stimulated by anti-CD3 antibody in vivo . ITK degrader 1 also shows good plasma exposure levels [1] .
Molecular Weight:
943.02
Purity:
0.98