Varenicline
Code | Size | Price |
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TAR-T4246L-100mg | 100mg | Enquire | |||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||
Special offer! Add £1 to your order to get a TargetMol CCK-8 Kit. Read more here. |
Quantity:
TAR-T4246L-50mg | 50mg | Enquire | |||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||
Special offer! Add £1 to your order to get a TargetMol CCK-8 Kit. Read more here. |
Quantity:
Prices exclude any Taxes / VAT
Overview
Regulatory Status: RUO
Shipping:
cool pack
Storage:
-20°C
Images
Documents
Further Information
Bioactivity:
Varenicline (CP 526555) is a potent partial α4β2 nicotinic acetylcholine receptor (nAChR) agonist with an EC 50 value of 2.3 uM. Varenicline is a full agonist for α3β4 and α7 nAChRs with EC 50 values of 55 uM and 18 uM, respectively [1]. Varenicline is a nicotinic ligand based on the structure of cytisine, has the potential for smoking cessation treatment [2].
CAS:
249296-44-4
Molecular Weight:
211.268
Purity:
0.98
SMILES:
C1C2CNCC1c1cc3nccnc3cc21