GRK6-IN-2
Code | Size | Price |
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TAR-T61556-100mg | 100mg | Enquire | |||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||
Special offer! Add £1 to your order to get a TargetMol CCK-8 Kit. Read more here. |
Quantity:
TAR-T61556-50mg | 50mg | Enquire | |||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||
Special offer! Add £1 to your order to get a TargetMol CCK-8 Kit. Read more here. |
Quantity:
Prices exclude any Taxes / VAT
Overview
Regulatory Status: RUO
Shipping:
cool pack
Storage:
-20°C
Images
Documents
Further Information
Bioactivity:
GRK6-IN-2 (compound 10a) is a highly effective inhibitor of G protein-coupled receptor kinase 6 (GRK6) exhibiting an IC50 value of 120 nM. GRK6 is an essential kinase for the viability of multiple myeloma (MM) cells. Consequently, GRK6-IN-2 holds promise for further exploration in multiple myeloma research [1].
CAS:
2677786-27-3
Molecular Weight:
376.439
Purity:
0.98
SMILES:
CCc1cc(Nc2nc(N[C@@H](C)c3ccc(F)cc3)nc3ccccc23)n[nH]1