AGN 192870
Code | Size | Price |
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TAR-T61588-50mg | 50mg | £724.00 | |||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||
Special offer! Add £1 to your order to get a TargetMol CCK-8 Kit. Read more here. |
Quantity:
TAR-T61588-100mg | 100mg | £1,123.00 | |||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||
Special offer! Add £1 to your order to get a TargetMol CCK-8 Kit. Read more here. |
Quantity:
Prices exclude any Taxes / VAT
Overview
Regulatory Status: RUO
Shipping:
cool pack
Storage:
-20°C
Images
Documents
Further Information
Bioactivity:
AGN 192870 is a chemical compound that acts as a RAR neutral antagonist, inhibiting the activity of RARα, RARβ, and RARγ with Kd values of 147 nM, 33 nM, and 42 nM, respectively. It demonstrates IC50 values of 87 nM and 32 nM for RARα and RARγ, respectively. Additionally, AGN 192870 exhibits partial agonism towards RARβ.
CAS:
166977-57-7
Molecular Weight:
378.471
Purity:
0.98
SMILES:
CC1(C)CC=C(c2ccccc2)c2cc(ccc12)C#Cc1ccc(cc1)C(O)=O