GPR81 agonist 1
Code | Size | Price |
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TAR-T62656-50mg | 50mg | £1,364.00 | |||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||
Special offer! Add £1 to your order to get a TargetMol CCK-8 Kit. Read more here. |
Quantity:
TAR-T62656-100mg | 100mg | £1,990.00 | |||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||
Special offer! Add £1 to your order to get a TargetMol CCK-8 Kit. Read more here. |
Quantity:
Prices exclude any Taxes / VAT
Overview
Regulatory Status: RUO
Shipping:
cool pack
Storage:
-20°C
Images
Documents
Further Information
Bioactivity:
GPR81 agonist 1 is a highly selective and potent GPR81 agonist that acts in human (IC50: 58 nM) and mouse (IC50: 50 nM). GPR81 agonist 1 is more selective for GPR81 than GPR109a. GPR81 agonist 1 inhibits lipolysis in mice and does not cause skin flushing.
CAS:
1620992-67-7
Molecular Weight:
446.63
Purity:
0.98
SMILES:
C[C@H]1CC[C@@H](CC1)C(=O)Nc1nc(c(CC(=O)N2CCN(C)CC2)s1)-c1cccs1