AZ13705339 hemihydrate

TargetMol
Product Code: TAR-T72321
Supplier: TargetMol
CodeSizePrice
TAR-T72321-50mg50mg£752.00
Special offer! Add £1 to your order to get a TargetMol CCK-8 Kit. Read more here.
Quantity:
TAR-T72321-100mg100mg£1,099.00
Special offer! Add £1 to your order to get a TargetMol CCK-8 Kit. Read more here.
Quantity:
Prices exclude any Taxes / VAT

Overview

Regulatory Status: RUO
Shipping:
cool pack
Storage:
-20°C

Further Information

Bioactivity:
AZ13705339 hemihydrate is a highly potent and selective PAK1 inhibitor with IC 50 s of 0.33 nM and 59 nM for PAK1 and pPAK1, respectively. AZ13705339 hemihydrate has binding affinities to PAK1 and PAK2 , with K d s of 0.28 nM and 0.32 nM, respectively. AZ13705339 hemihydrate can be used in the research of cancers .
Molecular Weight:
638.77
Purity:
0.98
SMILES:
CCS(=O)(C1=C(N2CCN(C)CC2)C=CC(NC3=NC=C(F)C(N(C4=C(C)C=CC(CO)=C4)CC5=CC=CC=C5C#N)=N3)=C1)=O.CCS(=O)(C6=C(N7CCN(C)CC7)C=CC(NC8=NC=C(F)C(N(C9=C(C)C=CC(CO)=C9)CC%10=CC=CC=C%10C#N)=N8)=C6)=O.O