RGB-286638
Code | Size | Price |
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TAR-T73196-50mg | 50mg | £870.00 | |||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||
Special offer! Add £1 to your order to get a TargetMol CCK-8 Kit. Read more here. |
Quantity:
TAR-T73196-100mg | 100mg | £1,669.00 | |||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||
Special offer! Add £1 to your order to get a TargetMol CCK-8 Kit. Read more here. |
Quantity:
Prices exclude any Taxes / VAT
Overview
Regulatory Status: RUO
Shipping:
cool pack
Storage:
-20°C
Images
Documents
Further Information
Bioactivity:
RGB-286638 is a CDK inhibitor that inhibits the kinase activity of cyclin T1-CDK9 , cyclin B1-CDK1 , cyclin E-CDK2 , cyclin D1-CDK4 , cyclin E-CDK3 , and p35-CDK5 with IC 50 s of 1, 2, 3, 4, 5 and 5 nM, respectively ; also inhibits GSK-3β , TAK1, Jak2 and MEK1 , with IC 50 s of 3, 5, 50, and 54 nM.
CAS:
784210-87-3
Molecular Weight:
618.55
Purity:
0.98
SMILES:
Cl.Cl.O=C(NC1=CC=CC=2C=3NN=C(C=4C=CC(=CC4)CN5CCN(CCOC)CC5)C3C(=O)C12)NN6CCOCC6