PD 168368
Code | Size | Price |
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TAR-T8691-50mg | 50mg | £1,099.00 | |||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||
Special offer! Add £1 to your order to get a TargetMol CCK-8 Kit. Read more here. |
Quantity:
TAR-T8691-100mg | 100mg | £1,669.00 | |||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||
Special offer! Add £1 to your order to get a TargetMol CCK-8 Kit. Read more here. |
Quantity:
Prices exclude any Taxes / VAT
Overview
Regulatory Status: RUO
Shipping:
cool pack
Storage:
-20°C
Images
Documents
Further Information
Bioactivity:
PD 168368 is a potent, competitive, and selective neuromedin B receptor ( NMB-R ) antagonist with the K i of 15?45 nM [1]. PD 168368 is a dual antagonist of neuromedin B receptor ( NMBR; IC 50 =96 nM) / gastrin-releasing peptide receptor ( GRPR IC 50 =3500 nM) [2]. PD 168368 also is a mixed FPR1/FPR2/FPR3 agonist with EC 50 s of 0.57, 0.24, and 2.7 nM, respectively [3].
CAS:
204066-82-0
Formula:
C31H34N6O4
Molecular Weight:
554.64
Purity:
0.98
SMILES:
C[C@@](Cc1c[nH]c2ccccc12)(NC(=O)Nc1ccc(cc1)[N+]([O-])=O)C(=O)NCC1(CCCCC1)c1ccccn1