AT6
Code | Size | Price |
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TAR-T13561-100mg | 100mg | Enquire | |||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||
Special offer! Add £1 to your order to get a TargetMol CCK-8 Kit. Read more here. |
Quantity:
TAR-T13561-500mg | 500mg | Enquire | |||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||
Special offer! Add £1 to your order to get a TargetMol CCK-8 Kit. Read more here. |
Quantity:
Prices exclude any Taxes / VAT
Overview
Regulatory Status: RUO
Shipping:
cool pack
Storage:
-20°C
Images
Documents
Further Information
Bioactivity:
AT6 is a PROTAC AT1 analog which is a highly selective bromodomain (Brd4) degrader.
CAS:
2098836-50-9
Formula:
C48H58ClN9O7S3
Molecular Weight:
1004.68
Purity:
0.98
SMILES:
CC=1C2=C(N3C([C@H](CC(NCCOCCOCCSC([C@@H](C(=O)N4[C@H](C(NCC5=CC=C(C=C5)C6=C(C)N=CS6)=O)C[C@@H](O)C4)NC(C)=O)(C)C)=O)N=C2C7=CC=C(Cl)C=C7)=NN=C3C)SC1C
References
Gadd MS, et al. Structural basis of PROTAC cooperative recognition for selective protein degradation. Nat Chem Biol. 2017 May;13(5):514-521.