BMS-986020 sodium
| Code | Size | Price |
|---|
| TAR-T63439-500mg | 500mg | £1,388.00 | |||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||
| Special offer! Add £1 to your order to get a TargetMol CCK-8 Kit. Read more here. | |||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||
Quantity:
Prices exclude any Taxes / VAT
Overview
Regulatory Status: RUO
Shipping:
cool pack
Storage:
-20°C
Documents
Further Information
Bioactivity:
BMS-986020 sodium is a high-affinity lysophosphatidic acid receptor 1 (LPA1) antagonist that inhibits bile acids and phospholipid transport proteins, and inhibits BSEP (IC50: 4.8 uM), MRP4 (IC50: 6.2 uM) and MDR3 (IC50: 7.5 uM). BMS-986020 sodium showed potential for the study of idiopathic pulmonary fibrosis (IPF).
CAS:
1380650-53-2
Molecular Weight:
504.518
Purity:
0.98
SMILES:
[Na+].C[C@@H](OC(=O)Nc1c(C)noc1-c1ccc(cc1)-c1ccc(cc1)C1(CC1)C([O-])=O)c1ccccc1