PIK-294
| Code | Size | Price |
|---|
| SYN-1098-M100 | 100 mg | Enquire |
Quantity:
| SYN-1098-M001 | 1 mg | £133.00 |
Quantity:
| SYN-1098-M005 | 5 mg | £197.00 |
Quantity:
| SYN-1098-M010 | 10 mg | £350.00 |
Quantity:
| SYN-1098-M050 | 50 mg | £1,053.00 |
Quantity:
Prices exclude any Taxes / VAT
Overview
Regulatory Status: RUO
Shipping:
-20°C
Documents
Further Information
Alternate Names/Synonyms:
PIK294
Appearance:
Solid.
CAS:
900185-02-6
EClass:
32160000
Form (Short):
liquid
InChi:
InChI=1S/C28H23N7O2/c1-16-7-3-4-12-21(16)35-22(32-20-11-5-8-17(2)23(20)28(35)37)14-34-27-24(26(29)30-15-31-27)25(33-34)18-9-6-10-19(36)13-18/h3-13,15,36H,14H2,1-2H3,(H2,29,30,31)
InChiKey:
WFSLJOPRIJSOJR-UHFFFAOYSA-N
Long Description:
Chemical. CAS: 900185-02-6. Formula: C28H23N7O2. MW: 489.5. PIK-294 is a PI3 Kinase inhibitor that is 20- to 60-fold more potent than the parent compound, PIK-293. It is one of the most potent p110delta-selective inhibitors that has been reported, with an IC(50) of 10nM.
Molecular Formula:
C28H23N7O2
Molecular Weight:
489.5
Package Type:
Plastic Vial
Product Description:
PIK-294 is a PI3 Kinase inhibitor that is 20- to 60-fold more potent than the parent compound, PIK-293. It is one of the most potent p110delta-selective inhibitors that has been reported, with an IC(50) of 10nM.
Purity:
>95%
Solubility Chemicals:
Soluble in DMSO. Slightly soluble (<1mg/ml) in ethanol.
Transportation:
Non-hazardous
UNSPSC Category:
Protein Kinase Modulators
UNSPSC Number:
12352200
Use & Stability:
Stable for at least 2 years after receipt when stored at -20°C.
References
A pharmacological map of the PI3-K family defines a role for p110alpha in insulin signaling: Z.A. Knight, et al.; Cell 125, 733 (2006)
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